Description
Arimistane + Enclomiphene
Arimistane + Enclomiphene liquid is offered as 16,5mg Arimistane + 16.5mg Enclomiphene per liquid vial, totaling 33mg per vial or 1000mg in total.
Arimistane
Arimistane is an aromatase inhibitor which implies a reduction in the production of estrogen. Aromatase inhibitors are bound to the catalytic site, where they are transformed into electrophilic intermediates that become irreversibly attached to the enzyme, blocking its activity. These inhibitors have distinct advantages in compound design because they are highly enzyme-specific, produce prolonged inhibition, and exhibit minimal toxicities. Studies show that Arimistane as an aromatase inhibitor effectively delays epiphysial maturation in young subjects and improves testosterone levels in adult subjects by suppressing the production of estrogen.
| Arimistane Capsules | |
| CAS Number | 1420-49-1 |
| Molar Mass | 284.17g.mol-1 |
| Chemical Formula | C19H24O2 |
| IUPAC Name | (8R,9S,10R,13S,14S)-10,13-dimethyl-2,8,9,11,12,14,15,16-octahydro-1H-cyclopenta[a]phenanthrene-7,17-dione |
Enclomiphene
Enclomiphene is being studied for its potential to increase serum total testosterone levels while maintaining sperm counts in the normal range in men with secondary hypogonadism.
Enclomiphene is thus a powerful estrogen receptor (ER) modulator. It acts as an ER antagonist in humans, sheep, and rabbits and an ER agonist in rats. Enclomiphene works by inhibiting the binding of 17beta-estradiol in isolated rabbit uterus. It decreases E2-induced inhibition of follicle-stimulating hormone (FSH) secretion in primary sheep pituitary cells in a concentration-dependent manner. Enclomiphene (0.25 and 0.5 mg/animal) inhibits spermatogenesis and decreases serum luteinizing hormone (LH) and testosterone levels in intact or castrated rats. Formulations containing clomiphene have been used in the treatment of ovarian dysfunction. In addition, this compound may bind to estrogen receptors in breast cancer cells, resulting in the inhibition of estrogen-stimulated proliferation in susceptible cell populations.
| Enclomiphene | |
| CAS Number | 7599-79-3 |
| Molar Mass | 598.1g.mol-1 |
| Chemical Formula | C32H36ClNO8 |
| IUPAC Name | 2-[4-[(E)-2-chloro-1,2-diphenylethenyl]phenoxy]-N,N-diethylethanamine;2-hydroxypropane-1,2,3-tricarboxylic acid |
Cai Spence –
Great product!
Wyatt Gamble –
Very good for hormone balance. Wish I discovered this blend earlier.
Kevin Wyatt –
Effective results but delivery was slower than expected.
Gabriel Zimmerman –
Life-changing powerhouse of a combo. Highly recommend